Ramucirumab

The approval was based on the results of the REGARD trial, a phase III, international, randomized, double-blind, placebo-controlled study, that evaluated the safety and efficacy of ramucirumab combinated with best supportive care versus placebo.[11] In December 2014, the FDA approved ramucirumab in combination with docetaxel for treatment of metastatic non-small-cell lung carcinoma (NSCLC) with disease progression during or after first-line platinum-containing chemotherapy.[12] In April 2015, ramucirumab was approved by FDA for the treatment of patients with metastatic colorectal cancer (mCRC) with disease progression on or after prior therapy with bevacizumab, oxaliplatin, and fluoropyrimidine.In September 2013, the manufacturer Eli Lilly announced that its phase III study for ramucirumab failed to hit its primary endpoint on progression-free survival among women with metastatic breast cancer.[19] Between 2016 and 2018, 26 hospitals in Italy conducted a multicentre, randomised, double-blind, placebo-controlled, phase II trial to evaluate the safety and effectiveness of the anti-VEGFR-2 antibody ramucirumab combined with gemcitabine in patients with pretreated  pleural mesothelioma.
Monoclonal antibodyTargetVEGFR2Drugs.comMedlinePlusLicense dataDailyMedRoutes ofadministrationIntravenous infusionDrug classAntineoplastic agentsATC codeL01FG02Legal status ℞-only℞-onlyPharmacokineticMetabolismproteasesElimination half-lifeCAS NumberDrugBankChemSpiderFormulaMolar massImClone Systemsphage display libraryindicatedcavitationdiarrheaplacebohyponatraemiasodiumpaclitaxeldocetaxelirinotecanVEGF-AVEGF-CVEGF-DangiogenesisFood and Drug Administrationgastricadenocarcinomafluoropyrimidineplatinum-containing chemotherapynon-small-cell lung carcinomacolorectal cancerbevacizumaboxaliplatinfolinic acid5-fluorouracilFOLFIRIhepatocellular carcinomaalpha fetoproteinsorafenibrandomizeddouble-blindplacebo-controlledoverall survivalEli Lillyprogression-free survivalbreast cancerliver cancerurothelial carcinomaHealth CanadaEuropean Medicines AgencyClinicalTrials.govTargeted cancer therapymonoclonal antibodiesReceptor tyrosine kinaseHER1/EGFRCetuximabPanitumumabHER2/neuPertuzumabTrastuzumab+hyaluronidaseTrastuzumab emtansineTrastuzumab deruxtecanZanidatamabCatumaxomabEdrecolomabLeukemialymphomalymphoidGlofitamabElranatamabMosunetuzumabIbritumomabObinutuzumabOfatumumabRituximabTositumomabBrentuximabAlemtuzumabmyeloidGemtuzumab ozogamicinAmivantamabAtezolizumabAvelumabAxatilimabBelantamab mafodotinBermekimabBlinatumomabCemiplimabCosibelimabDaratumumabDinutuximab betaDostarlimabDurvalumabElotuzumabEnfortumab vedotinEpcoritamabInotuzumab ozogamicinIpilimumabIsatuximabLoncastuximab tesirineMirvetuximab soravtansineMogamulizumabMoxetumomab pasudotoxNaxitamabNecitumumabNivolumab+relatlimabOlaratumabOportuzumab monatoxPembrolizumabPolatuzumab vedotinRetifanlimabSacituzumab govitecanSerplulimabSugemalimabTafasitamabTalquetamabTarlatamabTeclistamabTislelizumabTisotumab vedotinToripalimabTremelimumabZenocutuzumabZolbetuximabTyrosine kinase inhibitorsAfatinibAumolertinibBrigatinibDacomitinibErlotinibGefitinibIcotinibLazertinibMobocertinibOlmutinibOsimertinibRociletinibVandetanibLapatinibNeratinibTucatinibDabrafenibEncorafenibTovorafenibVemurafenibRTK class IIIAvapritinibAxitinibMasitinibPazopanibRipretinibSunitinibToceranibLestaurtinibGilteritinibCediranibFruquintinibLenvatinibNintedanibRegorafenibSemaxanibTivozanibAlectinibCeritinibCrizotinibEnsartinibLorlatinibEntrectinibFutibatinibInfigratinibLarotrectinibPemigatinibPralsetinibRepotrectinibSelpercatinibCabozantinibCapmatinibNon-receptorbcr-ablAsciminibBosutinibDasatinibImatinibNilotinibPonatinibRadotinibJanus kinaseBaricitinibFedratinibFilgotinibMomelotinibPacritinibRuxolitinibBinimetinibCobimetinibSelumetinibTrametinibBruton'sAcalabrutinibIbrutinibOrelabrutinibPirtobrutinibZanubrutinibfusion proteinAfliberceptproapoptoticprohibitinAdipotideexotoxinDenileukin diftitoxmTOR inhibitorsEverolimusRidaforolimusSirolimusTemsirolimushedgehogGlasdegibSonidegibVismodegibCDK inhibitorsAbemaciclibDalpiciclibPalbociclibRibociclibTrilaciclibAdagrasibSotorasibPi3K inhibitorsAlpelisibCopanlisibDuvelisibIdelalisibInavolisibParsaclisibRevumenibFibroblast growth factor receptorErdafitinibMidostaurinOdronextamabPexidartinibQuizartinibTebentafuspTepotinibTunlametinibVenetoclaxAdecatumumabAscrinvacumabCixutumumabConatumumabDrozitumabDuligotumabDusigitumabEnoticumabFigitumumabFlanvotumabGanitumabGlembatumumab vedotinIntetumumabIratumumabIstiratumabIcrucumabLexatumumabLucatumumabMapatumumabNarnatumabNesvacumabPatritumabPritumumabRadretumabRilotumumabRobatumumabSeribantumabTarextumabTeprotumumabTovetumabVantictumabVotumumabZalutumumabAbagovomabAltumomab pentetateAnatumomab mafenatoxArcitumomabBectumomabCapromab pendetideDetumomabIbritumomab tiuxetanIgovomabLilotomabMinretumomabMitumomabNacolomab tafenatoxNaptumomab estafenatoxOregovomabPemtumomabRacotumomabSatumomab pendetideSolitomabTaplitumomab paptoxNofetumomab merpentanPintumomabTenatumomabChimericAmatuximabBavituximabBrentuximab vedotinCarotuximabDerlotuximab biotinDinutuximabEcromeximabEnsituximabFutuximabGirentuximabIndatuximab ravtansineMargetuximabSiltuximabUblituximabHumanizedAbituzumabBivatuzumab mertansineBrontictuzumabCantuzumab mertansineCantuzumab ravtansineCirmtuzumabCitatuzumab bogatoxClivatuzumab tetraxetanCofetuzumab pelidotinDacetuzumabDemcizumabDalotuzumabDatopotamab deruxtecanDenintuzumab mafodotinEmactuzumabEmibetuzumabEnoblituzumabEtaracizumabFarletuzumabFiclatuzumabFlotetuzumabImgatuzumabLabetuzumabLifastuzumab vedotinLintuzumabLorvotuzumab mertansineLumretuzumabMatuzumabMilatuzumabNimotuzumabOcaratuzumabOtlertuzumabOnartuzumabParsatuzumabPinatuzumab vedotinRosmantuzumabRovalpituzumab tesirineSibrotuzumabSimtuzumabSofituzumab vedotinTacatuzumab tetraxetanTigatuzumab+deruxtecan+emtansineTucotuzumab celmoleukinVandortuzumab vedotinVanucizumabVeltuzumabVorsetuzumab mafodotinRat/mouse hybridErtumaxomabDepatuxizumab mafodotinDuvortuxizumabOntuxizumabWHO-EMWithdrawnClinical trialsMonoclonalsBurosumabDenosumabBlosozumabRomosozumabMusculoskeletalStamulumabCirculatoryAbelacimabAlirocumabBentracimabEvinacumabEvolocumabInclacumabMarstacimabOrticumabRinucumabBiciromabImciromabAbciximabVolociximabAlacizumab pegolRanibizumabBococizumabBrolucizumabCaplacizumabConcizumabEmicizumabFaricimabIdarucizumabRalpancizumabTadocizumabNeurologicAnti-amyloid drugsAducanumabDonanemabGantenerumabLecanemabErenumabFasinumabFulranumabOpicinumabBapineuzumabCrenezumabEptinezumabFremanezumabGalcanezumabOzanezumabPonezumabRefanezumabSemorinemabSolanezumabTanezumabAngiogenesis inhibitorGrowth factorBimagrumabTrevogrumabDomagrozumabLandogrozumabGrowth factor receptormodulatorsAngiopoietinAngiopoietin 1Angiopoietin 4Angiopoietin 2RebastinibAxokineEGF (ErbB)EGF(ErbB1/HER1)AmphiregulinBetacellulinEGF (urogastrone)EpigenEpiregulinHeparin-binding EGF-like growth factor (HB-EGF)MuroderminNepiderminTransforming growth factor alpha (TGFα)CanertinibGrandininErbB2/HER2MubritinibErbB3/HER3Neuregulins (heregulins)6 (neuroglycan C)ErbB4/HER42 (bFGF)10 (KGF2)TraferminPaliferminSpriferminFGF15/19HGF (c-Met)FosgonimetonHepatocyte growth factorDihexa (PNB-0408)ForetinibTivantinibVolitinibTelisotuzumab vedotindes(1-3)IGF-1Insulin-like growth factor-1 (somatomedin C)IGF-1 LR3Insulin-like growth factor-2 (somatomedin A)InsulinMecaserminMecasermin rinfabateLinsitinibTrofinetideLNGF (p75NTR)BNN-20BNN-27CenegerminDHEA-SDexamethasoneTestosteroneFrunevetmabBecaplerminPlatelet-derived growth factorCrenolanibMotesanibRET (GFL)GFRα1Glial cell line-derived neurotrophic factor (GDNF)GFRα2Neurturin (NRTN)GFRα3Artemin (ARTN)GFRα4Persephin (PSPN)SCF (c-Kit)AncestimStem cell factorAmitriptylineTavilermide4'-DMA-7,8-DHF7,8-DHF7,8,3'-THFDeoxygeduninDeprenylDiosmetinLM22A-4N-AcetylserotoninNorwogonin (5,7,8-THF)ANA-12Cyclotraxin BGossypetin (3,5,7,8,3',4'-HHF)Placental growth factor (PGF)D (FIGF)PegaptanibAdrenomedullinColony-stimulating factorsConnective tissue growth factor (CTGF)EphrinsErythropoietinGlucose-6-phosphate isomerase (GPI; PGI, PHI, AMF)Glia maturation factor (GMF)Hepatoma-derived growth factor (HDGF)InterleukinsT-cell growth factorsLeukemia inhibitory factor (LIF)Macrophage-stimulating protein (MSP; HLP, HGFLP)Midkine (NEGF2)Migration-stimulating factor (MSF; PRG4)OncomodulinPituitary adenylate cyclase-activating peptide (PACAP)PleiotrophinRenalaseThrombopoietinWnt signaling proteinsCerebrolysinEli Lilly and CompanyCorporatedirectorsJohn C. LechleiterRalph AlvarezSir Winfried BischoffMichael L. EskewMartin S. FeldsteinAlfred G. GilmanKaren N. HornDouglas R. OberhelmanKathi P. SeifertAdcircaAlimtaAmyvidBamlanivimabBaqsimiBasaglarCialisCymbaltaCyramzaEmgalityErbituxEtesevimabEvistaForteoGemzarGlucagonGlyxambiHumalogHumatropeHumulinJardianceJaypircaJentaduetoKisunlaLyumjevOlumiantPortrazzaProzacRetevmoReyvowStratteraSymbyaxSynjardyTradjentaTrijardyTrulicityVerzenioXigrisZyprexa