Retifanlimab

Retifanlimab, sold under the brand name Zynyz, is an anti-cancer medication used for the treatment of Merkel cell carcinoma.[1][2][3][4][5] Retifanlimab is indicated for the treatment of adults with metastatic or recurrent locally advanced Merkel cell carcinoma.[1][2][6] The US Food and Drug Administration (FDA) evaluated the safety and efficacy of retifanlimab based on PODIUM-201 (NCT03599713), an open-label, multiregional, single-arm study evaluating 65 participants with metastatic or recurrent locally advanced MCC who had not received prior systemic therapy for advanced disease.[2] The FDA granted the application for retifanlimab priority review, fast track, and orphan drug designations.[7] The applicant for this medicinal product is Incyte Biosciences Distribution B.V.[7] Retifanlimab is the international nonproprietary name.
Monoclonal antibodyHumanizedTargetProgrammed cell death protein 1Drugs.comMedlinePlusLicense dataDailyMedRoutes ofadministrationIntravenousATC codeL01FF10Legal status℞-onlyCAS NumberDrugBankFormulaMolar massanti-cancer medicationMerkel cell carcinomaprogrammed death receptor-1indicatedFood and Drug Administrationpriority reviewfast trackorphan drugCommittee for Medicinal Products for Human UseEuropean Medicines Agencyinternational nonproprietary namepublic domainWorld Health OrganizationClinicalTrials.govTargeted cancer therapyantineoplastic agentsmonoclonal antibodiesReceptor tyrosine kinaseHER1/EGFRCetuximabPanitumumabHER2/neuPertuzumabTrastuzumab+hyaluronidaseTrastuzumab emtansineTrastuzumab deruxtecanZanidatamabCatumaxomabEdrecolomabVEGF-ABevacizumabLeukemialymphomalymphoidGlofitamabElranatamabMosunetuzumabIbritumomabObinutuzumabOfatumumabRituximabTositumomabBrentuximabAlemtuzumabmyeloidGemtuzumab ozogamicinAmivantamabAtezolizumabAvelumabAxatilimabBelantamab 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