Tislelizumab

[12] In the EU, tislelizumab is indicated for the treatment of adults with unresectable, locally advanced or metastatic esophageal squamous cell carcinoma after prior platinum-based chemotherapy.[5] In November 2024, the European Commission expanded the indication of tislelizumab for use alongside platinum- and fluoropyrimidine-based chemotherapy to treat people with HER2-negative locally advanced unresectable or metastatic gastric or gastroesophageal junction adenocarcinoma; and, in combination with platinum-based chemotherapy, for those with unresectable, locally advanced or metastatic esophageal squamous cell carcinoma.[5][13] In the US, tislelizumab is indicated for the treatment of adults with unresectable or metastatic esophageal squamous cell carcinoma after prior systemic chemotherapy that did not include a PD-(L)1 inhibitor;[4] and, in combination with platinum and fluoropyrimidine-based chemotherapy, it is indicated for the first-line treatment of adults with unresectable or metastatic HER2-negative gastric or gastroesophageal junction adenocarcinoma whose tumors express PD-L1.[4] Adverse effects include anemia, leukopenia, thrombocytopenia, nausea, increased aspartate transaminase (AST), neutropenia, fatigue, decreased appetite, vomiting, musculoskeletal pain, constipation, hypoproteinemia and rash.[7][22] In November 2024, the European Medicines Agency expanded the indication of tislelizumab as part of a first-line combination treatment for adults with advanced gastric or esophageal cancer.
Fab fragmentextracellular domainMonoclonal antibodyHumanizedTargetDrugs.comMedlinePlusLicense dataDailyMedPregnancycategoryRoutes ofadministrationIntravenousDrug classAntineoplastic agentATC codeL01FF09Legal status℞-onlyCAS NumberDrugBankChemSpideranti-cancer medicationprogrammed death receptor-1BeiGeneindicatedHodgkin lymphomaurothelial carcinomachemotherapygastroesophageal junction adenocarcinomasquamous cell carcinomaanemialeukopeniathrombocytopenianauseaaspartate transaminaseneutropeniafatiguehypoproteinemiarespiratory infectionfailurehepatic injuryelimination half-lifepembrolizumabnivolumaburothelial cancerhepatocellular carcinomaEuropean Medicines Agencyinternational nonproprietary nameFood and Drug AdministrationClinicalTrials.govWorld Health OrganizationTargeted cancer therapyantineoplastic agentsmonoclonal antibodiesReceptor tyrosine kinaseHER1/EGFRCetuximabPanitumumabHER2/neuPertuzumabTrastuzumab+hyaluronidaseTrastuzumab emtansineTrastuzumab deruxtecanZanidatamabCatumaxomabEdrecolomabVEGF-ABevacizumabLeukemialymphomalymphoidGlofitamabElranatamabMosunetuzumabIbritumomabObinutuzumabOfatumumabRituximabTositumomabBrentuximabAlemtuzumabmyeloidGemtuzumab ozogamicinAmivantamabAtezolizumabAvelumabAxatilimabBelantamab mafodotinBermekimabBlinatumomabCemiplimabCosibelimabDaratumumabDinutuximab betaDostarlimabDurvalumabElotuzumabEnfortumab vedotinEpcoritamabInotuzumab ozogamicinIpilimumabIsatuximabLoncastuximab tesirineMirvetuximab soravtansineMogamulizumabMoxetumomab pasudotoxNaxitamabNecitumumab+relatlimabOlaratumabOportuzumab monatoxPolatuzumab vedotinRamucirumabRetifanlimabSacituzumab govitecanSerplulimabSugemalimabTafasitamabTalquetamabTarlatamabTeclistamabTisotumab vedotinToripalimabTremelimumabZenocutuzumabZolbetuximabTyrosine kinase inhibitorsAfatinibAumolertinibBrigatinibDacomitinibErlotinibGefitinibIcotinibLazertinibMobocertinibOlmutinibOsimertinibRociletinibVandetanibLapatinibNeratinibTucatinibDabrafenibEncorafenibTovorafenibVemurafenibRTK class IIIAvapritinibAxitinibMasitinibPazopanibRipretinibSorafenibSunitinibToceranibLestaurtinibGilteritinibCediranibFruquintinibLenvatinibNintedanibRegorafenibSemaxanibTivozanibAlectinibCeritinibCrizotinibEnsartinibLorlatinibEntrectinibFutibatinibInfigratinibLarotrectinibPemigatinibPralsetinibRepotrectinibSelpercatinibCabozantinibCapmatinibNon-receptorbcr-ablAsciminibBosutinibDasatinibImatinibNilotinibPonatinibRadotinibJanus kinaseBaricitinibFedratinibFilgotinibMomelotinibPacritinibRuxolitinibBinimetinibCobimetinibSelumetinibTrametinibBruton'sAcalabrutinibIbrutinibOrelabrutinibPirtobrutinibZanubrutinibfusion proteinAfliberceptproapoptoticprohibitinAdipotideexotoxinDenileukin diftitoxmTOR inhibitorsEverolimusRidaforolimusSirolimusTemsirolimushedgehogGlasdegibSonidegibVismodegibCDK inhibitorsAbemaciclibDalpiciclibPalbociclibRibociclibTrilaciclibAdagrasibSotorasibPi3K inhibitorsAlpelisibCopanlisibDuvelisibIdelalisibInavolisibParsaclisibRevumenibFibroblast growth factor receptorErdafitinibMidostaurinOdronextamabPexidartinibQuizartinibTebentafuspTepotinibTunlametinibVenetoclaximmune systemImmunosuppressionAbrilumabAdalimumabAnifrolumabAtorolimumabBelimumabBleselumabBrodalumabCamidanlumab tesirineCarlumabDupilumabEldelumabEmapalumabFresolimumabGolimumabIanalumabLanadelumabLenzilumabLerdelimumabLirentelimabLirilumabMavrilimumabMetelimumabMorolimumabNamilumabOleclumabOxelumabPamrevlumabPlaculumabRelatlimabSarilumabSifalimumabTabalumabTezepelumabUlocuplumabVarlilumabUrelumabBertilimumabZanolimumabNivolumab/relatlimabAfelimomabElsilimomabFaralimomabGavilimomabInolimomabMaslimomabNerelimomabOdulimomabTelimomab aritoxVepalimomabZolimomab aritoxChimericAndecaliximabBasiliximabClenoliximabGaliximabGomiliximabInfliximabKeliximabLumiliximabPriliximabTeneliximabVapaliximabApolizumabAselizumabBenralizumabCamrelizumabCedelizumabCertolizumab pegolCrizanlizumabDaclizumabEculizumabEfalizumabEpratuzumabErlizumabEtrolizumabFontolizumabFrexalimabInebilizumabItolizumabLampalizumabLetolizumabLigelizumabLulizumab pegolMepolizumabNatalizumabOcrelizumabOmalizumabOzoralizumabPascolizumabPateclizumabPexelizumabPidilizumabPlozalizumabPRO 140QuilizumabRavulizumabReslizumabRontalizumabRovelizumabRuplizumabSamalizumabSatralizumabSiplizumabSpartalizumabTalizumabTeplizumabTocilizumabToralizumabTregalizumabVatelizumabVedolizumabVisilizumabVobarilizumabTGN1412IbalizumabOtelixizumabRozanolixizumabSutimlimabInterleukinBrazikumabBriakinumabCanakinumabFezakinumabFletikumabGuselkumabSecukinumabSirukumabTralokinumabUstekinumabAnrukinzumabBimekizumabClazakizumabGevokizumabIxekizumabMirikizumabLebrikizumabOlokizumabPerakizumabRisankizumabSpesolimabTildrakizumabLokivetmablesionsBesilesomabFanolesomabLemalesomabSulesomabWHO-EMWithdrawnClinical trials