Alemtuzumab

Alemtuzumab, sold under the brand names Campath and Lemtrada among others, is a medication used to treat chronic lymphocytic leukemia and multiple sclerosis.[11] However the low-to-moderate levels of evidence in the included, existing studies were noted and the need for larger high-quality randomised, double-blind, controlled trials comparing mono or combination therapy with alemtuzumab was highlighted.[6] In November 2018, the US Food and Drug Administration (FDA) issued a safety announcement[12] warning about rare but serious instances of stroke and blood vessel wall tears in multiple sclerosis patients who have received Lemtrada (alemtuzumab), mostly occurring within one day of initiating treatment and leading in some cases to permanent disability and even death.[15] The Summary of Product Characteristics provided in the electronic Medicines Compendium [eMC [16]] further lists common and uncommon adverse reactions that have been reported for Lemtrada, which include serious opportunistic nocardial infections and cytomegalovirus syndrome.[20][21] Cases of multiple sclerosis reactivation/relapse have also been reported[22] Alemtuzumab is a recombinant DNA-derived humanized IgG1 kappa monoclonal antibody that is directed against the cell surface glycoprotein CD52.[31] A 2009 retrospective study of alemtuzumab (10 mg IV weekly) in 20 patients (no controls) with severe steroid-resistant acute intestinal graft-versus-host disease after allogeneic hematopoietic stem cell transplantation (HSCT) demonstrated improvement.
Monoclonal antibodyHumanizedTargetDrugs.comMedlinePlusLicense dataDailyMedPregnancycategoryRoutes ofadministrationIntravenous infusionATC codeL04AG06Legal statusWARNINGPharmacokineticElimination half-lifeCAS NumberDrugBankChemSpiderChEMBLFormulaMolar massmedicationchronic lymphocytic leukemiamultiple sclerosisinjection into a veinlymphocytesstem cellsfludarabineantibody-dependent cell-mediated cytotoxicityFood and Drug AdministrationEuropean Medicines Agencyautoimmune diseaseregulatory T cellHerman WaldmannCambridge UniversityGreg Winterhypervariable loopsGenzymeBayer AGSanofioff-label useinternational nonproprietary namegraft-versus-host diseasehematopoietic stem cell transplantationcytomegalovirusaspergillosisBibcodeThe Wall Street JournalWorld Health Organizationcentral nervous systemSigns and symptomsAtaxiaDepressionDiplopiaDysarthriaDysphagiaFatigueIncontinenceNystagmusOptic neuritisUhthoff's phenomenonDiagnosis of multiple sclerosisMcDonald criteriaPoser criteriaClinically 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leukoencephalopathy with subcortical cystsCAMFAK syndromeCentral pontine myelinolysisMarchiafava–Bignami diseaseMitochondrial DNA depletion syndromeList of multiple sclerosis organizationsList of people with multiple sclerosisMultiple sclerosis drug pipelinePathophysiologyTargeted cancer therapyantineoplastic agentsmonoclonal antibodiesReceptor tyrosine kinaseHER1/EGFRCetuximabPanitumumabHER2/neuPertuzumabTrastuzumabTrastuzumab emtansineTrastuzumab deruxtecanZanidatamabCatumaxomabEdrecolomabVEGF-ABevacizumabLeukemialymphomalymphoidGlofitamabElranatamabMosunetuzumabIbritumomabObinutuzumabOfatumumabRituximabTositumomabBrentuximabmyeloidGemtuzumab ozogamicinAmivantamabAtezolizumabAvelumabAxatilimabBelantamab mafodotinBermekimabBlinatumomabCemiplimabCosibelimabDaratumumabDinutuximab betaDostarlimabDurvalumabElotuzumabEnfortumab vedotinEpcoritamabInotuzumab ozogamicinIpilimumabIsatuximabLoncastuximab tesirineMirvetuximab soravtansineMogamulizumabMoxetumomab 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