Nivolumab

[11] In May 2021, the FDA approved nivolumab for the treatment of completely resected esophageal or gastroesophageal junction cancer with residual pathologic disease after neoadjuvant chemoradiotherapy.[12] In August 2021, the FDA approved nivolumab for the adjuvant treatment of urothelial carcinoma who are at high risk of recurrence after undergoing radical resection.[23][24] In October 2024, the FDA approved nivolumab with platinum-doublet chemotherapy as neoadjuvant treatment, followed by single-agent nivolumab after surgery as adjuvant treatment, for adults with resectable (tumors ≥ 4 cm and/or node positive) non-small cell lung cancer (NSCLC) and no known epidermal growth factor receptor (EGFR) mutations or anaplastic lymphoma kinase (ALK) rearrangements.[27] In trials for melanoma, the following side effects occurred in more than 10% of subjects and more frequently than with chemotherapy alone: rash and itchy skin, cough, upper respiratory tract infections, and peripheral edema.Other clinically important side effects with less than 10% frequency were ventricular arrhythmia, inflammation of parts of the eye (iridocyclitis), infusion-related reactions,[vague] dizziness, peripheral and sensory neuropathy, peeling skin, erythema multiforme, vitiligo, and psoriasis.[28][29] Normally, certain cancer cells exploit the PD-1 pathway to shield themselves from the immune response by expressing programmed death-ligand 1 (PD-L1), which interacts with the PD-1 receptor and inhibits T-cell activation and proliferation.[38] In May 2016, the FDA approved nivolumab for the treatment of people with classical Hodgkin lymphoma who have relapsed or progressed after autologous hematopoietic stem cell transplantation and post-transplantation brentuximab vedotin.[39] In December 2017, the FDA granted approval to nivolumab for adjuvant treatment of melanoma with involvement of lymph nodes or for metastatic disease with complete resection.[40] In April 2018, the FDA granted approval to nivolumab in combination with ipilimumab for the first-line treatment of people with intermediate and poor risk advanced renal cell carcinoma.[42] In October 2020, the US Food and Drug Administration (FDA) approved the combination of nivolumab with ipilimumab for the first-line treatment of adults with malignant pleural mesothelioma (MPM) that cannot be removed by surgery.[16] In 2016, Bristol Myers Squibb announced the results of a clinical trial in which nivolumab failed to achieve its endpoint and was no better than traditional chemotherapy at treating newly diagnosed lung cancer.[47] Bristol Myers Squibb went on to attempt to gain approval for a combination therapy for lung cancer that included nivolumab and the company's older drug ipilimumab.[54] Phase I and II clinical trials have shown nivolumab as a promising and durable treatment option in melanoma as a single agent and in combination with ipilimumab.[55] In October 2022, the results of a phase III trial, CheckMate -76K, showed that Opdivo reduced the risk of death by 58% as an adjuvant therapy in participants with completely resected stage two melanoma, the most serious type of skin cancer.
Fab fragmentextracellular domainMonoclonal antibodyTargetDrugs.comMedlinePlusLicense dataDailyMedPregnancycategoryRoutes ofadministrationIntravenousDrug classImmunotherapyATC codeL01FF01Legal status ℞-only℞-onlyPharmacokineticElimination half-lifeCAS NumberDrugBankChemSpiderChEMBLFormulaMolar massbrand nameanti-cancer medicationcancermelanomalung cancermalignant pleural mesotheliomarenal cell carcinomaHodgkin lymphomahead and neck cancerurothelial carcinomacolon canceresophageal squamous cell carcinomaliver cancergastric cancerintravenouslypruritusastheniadyspneaarthralgiapyrexiablocks PD-1checkpoint inhibitorT cellsWorld Health Organization's List of Essential MedicinesChinese hamster ovary cellsindicatedmetastatic melanomaipilimumabBRAF inhibitornon-small cell lung cancerplatinum-based drugssmall cell lung canceranti-angiogenicbladder cancerplatinum-based chemotherapyFood and Drug Administrationchemoradiotherapyradical resectionrelatlimabcisplatingemcitabinethe 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vedotinVanucizumabVeltuzumabVorsetuzumab mafodotinRat/mouse hybridErtumaxomabDepatuxizumab mafodotinDuvortuxizumabOntuxizumabWHO-EMWithdrawnClinical trialsimmune systemImmunosuppressionAbrilumabAdalimumabAnifrolumabAtorolimumabBelimumabBleselumabBrodalumabCamidanlumab tesirineCarlumabDupilumabEldelumabEmapalumabFresolimumabGolimumabIanalumabLanadelumabLenzilumabLerdelimumabLirentelimabLirilumabMavrilimumabMetelimumabMorolimumabNamilumabOleclumabOxelumabPamrevlumabPlaculumabSarilumabSifalimumabTabalumabTezepelumabUlocuplumabVarlilumabUrelumabBertilimumabZanolimumabAfelimomabElsilimomabFaralimomabGavilimomabInolimomabMaslimomabNerelimomabOdulimomabTelimomab aritoxVepalimomabZolimomab aritoxAndecaliximabBasiliximabClenoliximabGaliximabGomiliximabInfliximabKeliximabLumiliximabPriliximabTeneliximabVapaliximabApolizumabAselizumabBenralizumabCamrelizumabCedelizumabCertolizumab 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