Dinutuximab

Dinutuximab beta is also used as a second line treatment for children with high-risk neuroblastoma; it was tested and is used with a longer and slower dosing regime, and is given on its own, although it may be combined with IL-2 if a stronger immune response is needed.[9] More than 25% of children taking these drugs experienced pain, fever, hives, vomiting, diarrhea, bone marrow suppression causing loss of platelets, red blood cells, white blood cells, and albumin, hypotension, electrolyte imbalance including low sodium, potassium, and calcium, elevated transaminases, infusion reactions, and capillary leak syndrome.[5] In clinical trials of dinutuximab, the maximum plasma concentration was 11.5 mcg/mL; the mean steady state volume distribution was 5.4 L; the clearance rate was 0.21 L/day; and the average half-life was 10 days.[5][10] The version of dinutuximab made by United Therapeutics, and marketed under the brand name Unituxin, is manufactured via industrial fermentation using a murine myeloma cell line, SP2/0.[11][12] Dinutuximab (originally called Ch14.18) was discovered by a group at University of California San Diego led by Alice Yu; this antibody and several others were brought into clinical trials funded by the National Cancer Institute.
Monoclonal antibodyChimericTargetDrugs.comMedlinePlusLicense dataDailyMedPregnancycategoryRoutes ofadministrationIntravenousATC codeL01FX06Legal status ℞-onlyWARNINGCAS NumberIUPHAR/BPSDrugBankChemSpiderChEMBLFormulaMolar massneuroblastomaneuroectodermalcentral nervous systemperipheral nervesgranulocyte-macrophage colony stimulating factorinterleukin-213-cis-retinoic acidmorphineinfusion reactiongranulocyte-macrophage colony-stimulating factorinfusion reactionsneuropathic painbone marrow suppressionelectrolyte imbalanceelevated transaminasescapillary leak syndromeglycolipidneuroectodermprenatal developmentcell-mediated cytotoxicitycomplement-dependent cytotoxicityindustrial fermentationChinese hamster ovary cellsMemorial Sloan KetteringHealth CanadaFood and Drug AdministrationEuropean Medicines AgencyTargeted cancer therapyantineoplastic agentsmonoclonal antibodiesReceptor tyrosine kinaseHER1/EGFRCetuximabPanitumumabHER2/neuPertuzumabTrastuzumab+hyaluronidaseTrastuzumab emtansineTrastuzumab deruxtecanZanidatamabCatumaxomabEdrecolomabVEGF-ABevacizumabLeukemialymphomalymphoidGlofitamabElranatamabMosunetuzumabIbritumomabObinutuzumabOfatumumabRituximabTositumomabBrentuximabAlemtuzumabmyeloidGemtuzumab ozogamicinAmivantamabAtezolizumabAvelumabAxatilimabBelantamab mafodotinBermekimabBlinatumomabCemiplimabCosibelimabDaratumumabDinutuximab betaDostarlimabDurvalumabElotuzumabEnfortumab vedotinEpcoritamabInotuzumab ozogamicinIpilimumabIsatuximabLoncastuximab tesirineMirvetuximab soravtansineMogamulizumabMoxetumomab pasudotoxNaxitamabNecitumumabNivolumab+relatlimabOlaratumabOportuzumab monatoxPembrolizumabPolatuzumab vedotinRamucirumabRetifanlimabSacituzumab govitecanSerplulimabSugemalimabTafasitamabTalquetamabTarlatamabTeclistamabTislelizumabTisotumab vedotinToripalimabTremelimumabZenocutuzumabZolbetuximabTyrosine kinase inhibitorsAfatinibAumolertinibBrigatinibDacomitinibErlotinibGefitinibIcotinibLazertinibMobocertinibOlmutinibOsimertinibRociletinibVandetanibLapatinibNeratinibTucatinibDabrafenibEncorafenibTovorafenibVemurafenibRTK class IIIAvapritinibAxitinibMasitinibPazopanibRipretinibSorafenibSunitinibToceranibLestaurtinibGilteritinibCediranibFruquintinibLenvatinibNintedanibRegorafenibSemaxanibTivozanibAlectinibCeritinibCrizotinibEnsartinibLorlatinibEntrectinibFutibatinibInfigratinibLarotrectinibPemigatinibPralsetinibRepotrectinibSelpercatinibCabozantinibCapmatinibNon-receptorbcr-ablAsciminibBosutinibDasatinibImatinibNilotinibPonatinibRadotinibJanus kinaseBaricitinibFedratinibFilgotinibMomelotinibPacritinibRuxolitinibBinimetinibCobimetinibSelumetinibTrametinibBruton'sAcalabrutinibIbrutinibOrelabrutinibPirtobrutinibZanubrutinibfusion proteinAfliberceptproapoptoticprohibitinAdipotideexotoxinDenileukin diftitoxmTOR inhibitorsEverolimusRidaforolimusSirolimusTemsirolimushedgehogGlasdegibSonidegibVismodegibCDK inhibitorsAbemaciclibDalpiciclibPalbociclibRibociclibTrilaciclibAdagrasibSotorasibPi3K inhibitorsAlpelisibCopanlisibDuvelisibIdelalisibInavolisibParsaclisibRevumenibFibroblast growth factor receptorErdafitinibMidostaurinOdronextamabPexidartinibQuizartinibTebentafuspTepotinibTunlametinibVenetoclaxAdecatumumabAscrinvacumabCixutumumabConatumumabDrozitumabDuligotumabDusigitumabEnoticumabFigitumumabFlanvotumabGanitumabGlembatumumab vedotinIntetumumabIratumumabIstiratumabIcrucumabLexatumumabLucatumumabMapatumumabNarnatumabNesvacumabPatritumabPritumumabRadretumabRilotumumabRobatumumabSeribantumabTarextumabTeprotumumabTovetumabVantictumabVotumumabZalutumumabAbagovomabAltumomab pentetateAnatumomab mafenatoxArcitumomabBectumomabCapromab pendetideDetumomabIbritumomab tiuxetanIgovomabLilotomabMinretumomabMitumomabNacolomab tafenatoxNaptumomab estafenatoxOregovomabPemtumomabRacotumomabSatumomab pendetideSolitomabTaplitumomab paptoxNofetumomab merpentanPintumomabTenatumomabAmatuximabBavituximabBrentuximab vedotinCarotuximabDerlotuximab biotinEcromeximabEnsituximabFutuximabGirentuximabIndatuximab ravtansineMargetuximabSiltuximabUblituximabHumanizedAbituzumabBivatuzumab mertansineBrontictuzumabCantuzumab mertansineCantuzumab ravtansineCirmtuzumabCitatuzumab bogatoxClivatuzumab tetraxetanCofetuzumab pelidotinDacetuzumabDemcizumabDalotuzumabDatopotamab deruxtecanDenintuzumab mafodotinEmactuzumabEmibetuzumabEnoblituzumabEtaracizumabFarletuzumabFiclatuzumabFlotetuzumabImgatuzumabLabetuzumabLifastuzumab vedotinLintuzumabLorvotuzumab mertansineLumretuzumabMatuzumabMilatuzumabNimotuzumabOcaratuzumabOtlertuzumabOnartuzumabParsatuzumabPinatuzumab vedotinRosmantuzumabRovalpituzumab tesirineSibrotuzumabSimtuzumabSofituzumab vedotinTacatuzumab tetraxetanTigatuzumab+deruxtecan+emtansineTucotuzumab celmoleukinVandortuzumab vedotinVanucizumabVeltuzumabVorsetuzumab mafodotinRat/mouse hybridErtumaxomabDepatuxizumab mafodotinDuvortuxizumabOntuxizumabWHO-EMWithdrawnClinical trials