Tebentafusp

Tebentafusp, sold under the brand name Kimmtrak, is an anti-cancer medication used to treat uveal melanoma (eye cancer).[6] The most common side effects include cytokine release syndrome, rash, pyrexia (fever), pruritus (itching), fatigue (tiredness), nausea, chills, abdominal pain (stomach pain), edema (swelling), hypotension (low blood pressure), dry skin, headache, and vomiting, and abnormal liver blood tests.[6][7][9][10] Efficacy was evaluated in IMCgp100-202 (NCT03070392), a randomized, open-label, multicenter trial of 378 participants with metastatic uveal melanoma.[7] Participants with clinically significant cardiac disease or symptomatic, untreated brain metastases were excluded.[10] The trial was conducted at 58 sites across 14 countries including Australia, Belgium, Canada, France, Germany, Italy, the Netherlands, Poland, the Russian Federation, Spain, Switzerland, Ukraine, the United Kingdom, and the United States.
License dataDailyMedPregnancycategoryRoutes ofadministrationIntravenousATC codeL01XX75Legal status ℞-onlyWARNINGCAS NumberDrugBankanti-cancer medicationuveal melanomabispecific gp100 peptide-HLA-directed CD3 T cell engagerintravenous infusioncytokine release syndromepyrexiapruritusfatiguenauseaabdominal painhypotensionFood and Drug Administrationfirst-in-class medicationindicatedpembrolizumabipilimumabdacarbazineImmunocorepriority reviewbreakthrough therapyorphan drugCommittee for Medicinal Products for Human UseEuropean Medicines Agencypublic domainClinicalTrials.govchemotherapeutic agentsantineoplastic agentsM phasemicrotubuleVinca alkaloidsVinblastineVincristineVindesineVinflunineVinorelbineTaxanesCabazitaxelDocetaxelLarotaxelOrtataxelPaclitaxelTesetaxelEpothilonesIxabepiloneDNA replicationantimetabolitesS phaseFolic acidDihydrofolate reductase inhibitorAminopterinMethotrexatePemetrexedPralatrexateThymidylate synthase inhibitorRaltitrexedPurineAdenosine deaminase 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