Cetuximab

[6] However, subsequent studies[7] and clinical trials (NRG Oncology RTOG 1016[8] and De-ESCALaTE HPV[9]) suggested cetuximab was significantly inferior in overall and progression-free survival, when compared with cisplatin.[12] Further severe infusion reactions include but are not limited to: fevers, chills, rigors, urticaria, itchiness, rash, hypotension, nausea, vomiting, headache, shortness of breath, wheezing, angioedema, dizziness, anaphylaxis, and cardiac arrest.[18] Studies have indicated that detection of KRAS gene mutations helps physicians identify patients that are unlikely to respond to treatment with targeted EGFR inhibitors, including cetuximab and panitumumab.[medical citation needed] There is some evidence that colorectal tumors with the KRAS G13D mutation (glycine to aspartate at codon 13) respond to EGFR inhibition (specifically, with Cetuximab).[36] A 2020 phase III multicenter randomized controlled trial headed by University College London showed that adding cetuximab to perioperative chemotherapy worsened survival for colorectal cancer patients with operable liver metastases.[37] A multicenter, single arm, phase II study is being conducted that is designed to evaluate the efficacy and safety of cetuximab for the treatment of advanced (unresectable)/metastatic, chordoma.
Monoclonal antibodyChimericTargetEGF receptorDrugs.comLicense dataDailyMedPregnancycategoryRoutes ofadministrationIntravenousATC codeL01FE01Legal status ℞-onlyWARNINGPharmacokineticElimination half-lifeCAS NumberDrugBankChemSpiderChEMBLCompTox DashboardFormulaMolar massepidermal growth factor receptormedicationcolorectal cancerhead and neck cancerintravenous infusionindicatedFood and Drug Administrationradiation therapysquamous cell carcinomaHPV statuscisplatinacne-like rashrigorsurticariaitchinessanaphylaxishypomagnesemiapanitumumabgenetic testingWeizmann Institute of ScienceImcloneRhone-Poulenc-RorerEli Lilly and CompanyMerck KGaAintravenous therapyBiosimilarsImClone stock trading caseinsider tradingMartha StewartSamuel D. WaksalMerrill Lynchgastric cancerUniversity College LondonEuropean Medicines AgencyBibcodeTargeted cancer therapyantineoplastic agentsmonoclonal antibodiesReceptor tyrosine kinaseHER1/EGFRHER2/neuPertuzumabTrastuzumab+hyaluronidaseTrastuzumab emtansineTrastuzumab deruxtecanZanidatamabCatumaxomabEdrecolomabVEGF-ABevacizumabLeukemialymphomalymphoidGlofitamabElranatamabMosunetuzumabIbritumomabObinutuzumabOfatumumabRituximabTositumomabBrentuximabAlemtuzumabmyeloidGemtuzumab ozogamicinAmivantamabAtezolizumabAvelumabAxatilimabBelantamab mafodotinBermekimabBlinatumomabCemiplimabCosibelimabDaratumumabDinutuximab betaDostarlimabDurvalumabElotuzumabEnfortumab vedotinEpcoritamabInotuzumab ozogamicinIpilimumabIsatuximabLoncastuximab tesirineMirvetuximab soravtansineMogamulizumabMoxetumomab pasudotoxNaxitamabNecitumumabNivolumab+relatlimabOlaratumabOportuzumab monatoxPembrolizumabPolatuzumab vedotinRamucirumabRetifanlimabSacituzumab govitecanSerplulimabSugemalimabTafasitamabTalquetamabTarlatamabTeclistamabTislelizumabTisotumab vedotinToripalimabTremelimumabZenocutuzumabZolbetuximabTyrosine kinase inhibitorsAfatinibAumolertinibBrigatinibDacomitinibErlotinibGefitinibIcotinibLazertinibMobocertinibOlmutinibOsimertinibRociletinibVandetanibLapatinibNeratinibTucatinibDabrafenibEncorafenibTovorafenibVemurafenibRTK class IIIAvapritinibAxitinibMasitinibPazopanibRipretinibSorafenibSunitinibToceranibLestaurtinibGilteritinibCediranibFruquintinibLenvatinibNintedanibRegorafenibSemaxanibTivozanibAlectinibCeritinibCrizotinibEnsartinibLorlatinibEntrectinibFutibatinibInfigratinibLarotrectinibPemigatinibPralsetinibRepotrectinibSelpercatinibCabozantinibCapmatinibNon-receptorbcr-ablAsciminibBosutinibDasatinibImatinibNilotinibPonatinibRadotinibJanus kinaseBaricitinibFedratinibFilgotinibMomelotinibPacritinibRuxolitinibBinimetinibCobimetinibSelumetinibTrametinibBruton'sAcalabrutinibIbrutinibOrelabrutinibPirtobrutinibZanubrutinibfusion proteinAfliberceptproapoptoticprohibitinAdipotideexotoxinDenileukin diftitoxmTOR inhibitorsEverolimusRidaforolimusSirolimusTemsirolimushedgehogGlasdegibSonidegibVismodegibCDK inhibitorsAbemaciclibDalpiciclibPalbociclibRibociclibTrilaciclibAdagrasibSotorasibPi3K inhibitorsAlpelisibCopanlisibDuvelisibIdelalisibInavolisibParsaclisibRevumenibFibroblast growth factor receptorErdafitinibMidostaurinOdronextamabPexidartinibQuizartinibTebentafuspTepotinibTunlametinibVenetoclaxAdecatumumabAscrinvacumabCixutumumabConatumumabDrozitumabDuligotumabDusigitumabEnoticumabFigitumumabFlanvotumabGanitumabGlembatumumab vedotinIntetumumabIratumumabIstiratumabIcrucumabLexatumumabLucatumumabMapatumumabNarnatumabNesvacumabPatritumabPritumumabRadretumabRilotumumabRobatumumabSeribantumabTarextumabTeprotumumabTovetumabVantictumabVotumumabZalutumumabAbagovomabAltumomab pentetateAnatumomab mafenatoxArcitumomabBectumomabCapromab pendetideDetumomabIbritumomab tiuxetanIgovomabLilotomabMinretumomabMitumomabNacolomab tafenatoxNaptumomab estafenatoxOregovomabPemtumomabRacotumomabSatumomab pendetideSolitomabTaplitumomab paptoxNofetumomab merpentanPintumomabTenatumomabAmatuximabBavituximabBrentuximab vedotinCarotuximabDerlotuximab biotinDinutuximabEcromeximabEnsituximabFutuximabGirentuximabIndatuximab ravtansineMargetuximabSiltuximabUblituximabHumanizedAbituzumabBivatuzumab mertansineBrontictuzumabCantuzumab mertansineCantuzumab ravtansineCirmtuzumabCitatuzumab bogatoxClivatuzumab tetraxetanCofetuzumab pelidotinDacetuzumabDemcizumabDalotuzumabDatopotamab deruxtecanDenintuzumab mafodotinEmactuzumabEmibetuzumabEnoblituzumabEtaracizumabFarletuzumabFiclatuzumabFlotetuzumabImgatuzumabLabetuzumabLifastuzumab vedotinLintuzumabLorvotuzumab mertansineLumretuzumabMatuzumabMilatuzumabNimotuzumabOcaratuzumabOtlertuzumabOnartuzumabParsatuzumabPinatuzumab vedotinRosmantuzumabRovalpituzumab tesirineSibrotuzumabSimtuzumabSofituzumab vedotinTacatuzumab tetraxetanTigatuzumab+deruxtecan+emtansineTucotuzumab celmoleukinVandortuzumab vedotinVanucizumabVeltuzumabVorsetuzumab mafodotinRat/mouse hybridErtumaxomabDepatuxizumab mafodotinDuvortuxizumabOntuxizumabWHO-EMWithdrawnClinical trialsGrowth factor receptormodulatorsAngiopoietinAngiopoietin 1Angiopoietin 4Angiopoietin 2RebastinibEvinacumabAxokineEGF (ErbB)EGF(ErbB1/HER1)AmphiregulinBetacellulinEGF (urogastrone)EpigenEpiregulinHeparin-binding EGF-like growth factor (HB-EGF)MuroderminNepiderminTransforming growth factor alpha (TGFα)CanertinibGrandininErbB2/HER2MubritinibErbB3/HER3Neuregulins (heregulins)6 (neuroglycan C)ErbB4/HER42 (bFGF)10 (KGF2)TraferminPaliferminSpriferminBurosumabFGF15/19HGF (c-Met)FosgonimetonHepatocyte growth factorDihexa (PNB-0408)ForetinibTivantinibVolitinibTelisotuzumab vedotindes(1-3)IGF-1Insulin-like growth factor-1 (somatomedin C)IGF-1 LR3Insulin-like growth factor-2 (somatomedin A)InsulinMecaserminMecasermin rinfabateLinsitinibTrofinetideLNGF (p75NTR)BNN-20BNN-27CenegerminDHEA-SDexamethasoneTestosteroneFasinumabFrunevetmabFulranumabTanezumabBecaplerminPlatelet-derived growth factorCrenolanibMotesanibRET (GFL)GFRα1Glial cell line-derived neurotrophic factor (GDNF)GFRα2Neurturin (NRTN)GFRα3Artemin (ARTN)GFRα4Persephin (PSPN)SCF (c-Kit)AncestimStem cell factorAmitriptylineTavilermide4'-DMA-7,8-DHF7,8-DHF7,8,3'-THFDeoxygeduninDeprenylDiosmetinLM22A-4N-AcetylserotoninNorwogonin (5,7,8-THF)ANA-12Cyclotraxin BGossypetin (3,5,7,8,3',4'-HHF)Placental growth factor (PGF)D (FIGF)PegaptanibAlacizumab pegolRanibizumabAdrenomedullinColony-stimulating factorsConnective tissue growth factor (CTGF)EphrinsErythropoietinGlucose-6-phosphate isomerase (GPI; PGI, PHI, AMF)Glia maturation factor (GMF)Hepatoma-derived growth factor (HDGF)InterleukinsT-cell growth factorsLeukemia inhibitory factor (LIF)Macrophage-stimulating protein (MSP; HLP, HGFLP)Midkine (NEGF2)Migration-stimulating factor (MSF; PRG4)OncomodulinPituitary adenylate cyclase-activating peptide (PACAP)PleiotrophinRenalaseThrombopoietinWnt signaling proteinsCerebrolysinCorporatedirectorsJohn C. LechleiterRalph AlvarezSir Winfried BischoffMichael L. EskewMartin S. FeldsteinAlfred G. GilmanKaren N. HornDouglas R. OberhelmanKathi P. SeifertAdcircaAlimtaAmyvidBamlanivimabBaqsimiBasaglarCialisCymbaltaCyramzaEmgalityErbituxEtesevimabEvistaForteoGemzarGlucagonGlyxambiHumalogHumatropeHumulinJardianceJaypircaJentaduetoKisunlaLyumjevOlumiantPortrazzaProzacRetevmoReyvowStratteraSymbyaxSynjardyTradjentaTrijardyTrulicityVerzenioXigrisZyprexaMerck SeronoBisoprololCladribineEfalizumabGonadotropin preparationsHuman chorionic gonadotropinInterferon beta-1aLevothyroxineLuteinizing hormoneMetforminMitoxantroneSaizenSerostimTegafur/uracilMerck GroupSerono