Amivantamab

[5] The most common side effects include rash, infusion-related reactions, skin infections around the fingernails or toenails, muscle and joint pain, shortness of breath, nausea, fatigue, swelling in the lower legs or hands or face, sores in the mouth, cough, constipation, vomiting and changes in certain blood tests.[6] In March 2024, the FDA approved amivantamab, in combination with carboplatin and pemetrexed, for the first-line treatment of locally advanced or metastatic non-small cell lung cancer with epidermal growth factor receptor (EGFR) exon 20 insertion mutations, as detected by an FDA-approved test.[11] The FDA also granted traditional approval to amivantamab for adults with locally advanced or metastatic non-small cell lung cancer with epidermal growth factor receptor exon 20 insertion mutations, as detected by an FDA-approved test, whose disease has progressed on or after platinum-based chemotherapy.[15] The US Food and Drug Administration (FDA) approved amivantamab based on CHRYSALIS, a multicenter, non-randomized, open label, multicohort clinical trial (NCT02609776) which included participants with locally advanced or metastatic non-small cell lung cancer (NSCLC) with EGFR exon 20 insertion mutations.[6] In March 2024, the FDA approved amivantamab, in combination with carboplatin and pemetrexed, for the first-line treatment of locally advanced or metastatic non-small cell lung cancer with epidermal growth factor receptor (EGFR) exon 20 insertion mutations, as detected by an FDA-approved test.
Space-filling modelMonoclonal antibodyTargetEpidermal growth factor receptorDrugs.comMedlinePlusLicense dataDailyMedPregnancycategoryRoutes ofadministrationIntravenous infusionDrug classAntineoplasticATC codeL01FX18Legal status ℞-only℞-onlyCAS NumberDrugBankFormulaMolar massbispecific monoclonal antibodynon-small cell lung cancerepidermal growth factorMET receptorFood and Drug Administrationfirst-in-class medicationindicatedcarboplatinpemetrexedlazertinibnon-small-cell lung cancerCommittee for Medicinal Products for Human UseEuropean Medicines Agencyinternational nonproprietary nameosimertinibpublic domainWorld Health Organizationpublic domain materialClinicalTrials.govTargeted cancer therapyantineoplastic agentsmonoclonal antibodiesReceptor tyrosine kinaseHER1/EGFRCetuximabPanitumumabHER2/neuPertuzumabTrastuzumab+hyaluronidaseTrastuzumab emtansineTrastuzumab 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