Brolucizumab

Brolucizumab sold under trade name Beovu among others, is a humanized single-chain antibody fragment for the treatment of neovascular (wet) age-related macular degeneration (AMD).[7][8] Brolucizumab successfully completed phase III development in wet age-related macular degeneration (AMD) meeting the primary efficacy endpoint of non-inferiority to aflibercept in mean change in best corrected visual acuity (BCVA) from baseline to week 48.Furthermore, brolucizumab demonstrated superiority to aflibercept in key secondary endpoint measures of disease activity in wet age-related macular degeneration, a leading cause of blindness in two head-to-head pivotal Phase III studies.[9][10][11][12] In October 2019, Novartis announced that the US Food and Drug Administration (FDA) approved brolucizumab injection for the treatment of wet age-related macular degeneration.[16][17] In June 2020, the FDA approved an updated prescription label for brolucizumab that included additional safety information—specifically including the characterization of adverse events, retinal vasculitis and retinal vascular occlusion, as part of the spectrum of intraocular inflammation observed in HAWK (NCT02307682)[11] and HARRIER (NCT02434328)[12] clinical trials and noted in the original prescribing information.
Monoclonal antibodySingle-chain variable fragmentHumanizedTargetVascular endothelial growth factor ADrugs.comMedlinePlusLicense dataDailyMedPregnancycategoryRoutes ofadministrationIntravitrealATC codeS01LA06Legal status ℞-only℞-onlyCAS NumberIUPHAR/BPSDrugBankChemSpiderFormulaMolar massneovascular (wet) age-related macular degenerationendophthalmitisretinal detachmentvascular endothelial growth factorFood and Drug Administrationafliberceptvisual acuityocclusive retinal vasculitisInternational Nonproprietary NameUnited States Adopted NameKaposi sarcomaglioblastomaWayback MachineEuropean Medicines Agencypublic domainClinicalTrials.govAmerican Medical AssociationWorld Health OrganizationMonoclonalsBurosumabDenosumabBlosozumabRomosozumabMusculoskeletalStamulumabCirculatoryAbelacimabAlirocumabAscrinvacumabBentracimabEnoticumabEvinacumabEvolocumabIcrucumabInclacumabMarstacimabNesvacumabOrticumabRamucirumabRinucumabBiciromabImciromabChimericAbciximabVolociximabAlacizumab pegolBevacizumabRanibizumabBococizumabCaplacizumabConcizumabDemcizumabEmicizumabEtaracizumabFaricimabIdarucizumabRalpancizumabTadocizumabVanucizumabNeurologicAnti-amyloid drugsAducanumabDonanemabGantenerumabLecanemabErenumabFasinumabFulranumabOpicinumabBapineuzumabCrenezumabEptinezumabFremanezumabGalcanezumabOzanezumabPonezumabRefanezumabSemorinemabSolanezumabTanezumabAngiogenesis inhibitorGrowth factorBimagrumabTrevogrumabDomagrozumabLandogrozumabWHO-EMWithdrawnClinical trialsOphthalmologicalsvascular disorderneovascularisationAnecortavePegaptanibVerteporfinGrowth factor receptormodulatorsAngiopoietinAngiopoietin 1Angiopoietin 4Angiopoietin 2RebastinibAxokineEGF (ErbB)EGF(ErbB1/HER1)AmphiregulinBetacellulinEGF (urogastrone)EpigenEpiregulinHeparin-binding EGF-like growth factor (HB-EGF)MuroderminNepiderminTransforming growth factor alpha (TGFα)AfatinibBrigatinibCanertinibDacomitinibErlotinibGefitinibGrandininIcotinibLapatinibNeratinibOsimertinibVandetanibCetuximabDepatuxizumab mafodotinFutuximabImgatuzumabMatuzumabNecitumumabNimotuzumabPanitumumabZalutumumabErbB2/HER2ErtumaxomabPertuzumabTrastuzumabTrastuzumab deruxtecanTrastuzumab emtansineMubritinibTucatinibErbB3/HER3Neuregulins (heregulins)6 (neuroglycan C)DuligotumabPatritumabSeribantumabErbB4/HER42 (bFGF)10 (KGF2)SelpercatinibTraferminPaliferminSpriferminInfigratinibFGF15/19HGF (c-Met)FosgonimetonHepatocyte growth factorDihexa (PNB-0408)CabozantinibCapmatinibCrizotinibForetinibTivantinibVolitinibEmibetuzumabFiclatuzumabFlanvotumabOnartuzumabRilotumumabTelisotuzumab vedotindes(1-3)IGF-1Insulin-like growth factor-1 (somatomedin C)IGF-1 LR3Insulin-like growth factor-2 (somatomedin A)InsulinMecaserminMecasermin rinfabateLinsitinibCixutumumabDalotuzumabFigitumumabGanitumabRobatumumabTeprotumumabDusigitumabTrofinetideLNGF (p75NTR)BNN-20BNN-27CenegerminDHEA-SDexamethasoneTestosteroneFrunevetmabBecaplerminPlatelet-derived growth factorAvapritinibAxitinibCrenolanibImatinibLenvatinibMasitinibMotesanibNintedanibPazopanibRadotinibQuizartinibRipretinibSunitinibSorafenibToceranibOlaratumabTovetumabRET (GFL)GFRα1Glial cell line-derived neurotrophic factor (GDNF)GFRα2Neurturin (NRTN)GFRα3Artemin (ARTN)GFRα4Persephin (PSPN)SCF (c-Kit)AncestimStem cell factorDasatinibNilotinibAmitriptylineTavilermideEntrectinibLarotrectinibLestaurtinib4'-DMA-7,8-DHF7,8-DHF7,8,3'-THFDeoxygeduninDeprenylDiosmetinLM22A-4N-AcetylserotoninNorwogonin (5,7,8-THF)ANA-12Cyclotraxin BGossypetin (3,5,7,8,3',4'-HHF)Placental growth factor (PGF)D (FIGF)CediranibFruquintinibRegorafenibSemaxanibTivozanibAdrenomedullinColony-stimulating factorsConnective tissue growth factor (CTGF)EphrinsErythropoietinGlucose-6-phosphate isomerase (GPI; PGI, PHI, AMF)Glia maturation factor (GMF)Hepatoma-derived growth factor (HDGF)InterleukinsT-cell growth factorsLeukemia inhibitory factor (LIF)Macrophage-stimulating protein (MSP; HLP, HGFLP)Midkine (NEGF2)Migration-stimulating factor (MSF; PRG4)OncomodulinPituitary adenylate cyclase-activating peptide (PACAP)PleiotrophinRenalaseThrombopoietinWnt signaling proteinsCerebrolysin