Romosozumab

Romosozumab, sold under the brand name Evenity (/ɪˈvɛnɪti/ ih-VENN-ih-tee or with the pin-pen merger, /ɪˈvɪnɪti/ ih-VINN-ih-tee), is a medication used to treat osteoporosis.[14] Currently, the drug contains a FDA boxed warning on its labeling stating that it may increase the risk of heart attack, stroke and cardiovascular death and should not be used in patients who have had a heart attack or stroke within the previous year.[15] In a large real-world study, prescription of romosozumab was associated with less adverse cardiovascular events compared to other osteoanabolic therapies.[16] Romosozumab was approved for medical use in Japan in January 2019,[10] the United States in April 2019[10] and the European Union in December 2019.[19] The UK's National Institute for Health and Care Excellence (NICE) decided to recommend romosozumab for use in England and Wales.
Monoclonal antibodyHumanizedTargetSclerostinDrugs.comMedlinePlusLicense dataDailyMedPregnancycategoryATC codeM05BX06Legal status ℞-only℞-onlyCAS NumberDrugBankChemSpiderFormulaMolar masspin-pen mergerosteoporosisfractures of the spineinjection site reactionsheart attacksstrokeshumanized monoclonal antibodyFood and Drug Administrationfirst-in-class medicationdenosumabalendronateboxed warningChiroscienceCelltechNational Institute for Health and Care ExcellenceHealth CanadaEuropean Medicines AgencyAmerican Medical Associationbone diseasesBisphosphonatesNitrogenousAlendronic acidIbandronic acidIncadronic acidMinodronic acidNeridronic acidPamidronic acidRisedronic acidZoledronic acidEtidronic acidClodronic acidTiludronic acidBone morphogenetic proteinsDibotermin alfaEptotermin alfaIpriflavoneAluminium chlorohydrateStrontium ranelateCathepsin KOdanacatibParathyroid hormone-related proteinanaloguesAbaloparatideTeriparatideCalcitoninCalciumVitamin DMonoclonalsBurosumabBlosozumabMusculoskeletalStamulumabCirculatoryAbelacimabAlirocumabAscrinvacumabBentracimabEnoticumabEvinacumabEvolocumabIcrucumabInclacumabMarstacimabNesvacumabOrticumabRamucirumabRinucumabBiciromabImciromabChimericAbciximabVolociximabAlacizumab pegolBevacizumabRanibizumabBococizumabBrolucizumabCaplacizumabConcizumabDemcizumabEmicizumabEtaracizumabFaricimabIdarucizumabRalpancizumabTadocizumabVanucizumabNeurologicAnti-amyloid drugsAducanumabDonanemabGantenerumabLecanemabErenumabFasinumabFulranumabOpicinumabBapineuzumabCrenezumabEptinezumabFremanezumabGalcanezumabOzanezumabPonezumabRefanezumabSemorinemabSolanezumabTanezumabAngiogenesis inhibitorGrowth factorBimagrumabTrevogrumabDomagrozumabLandogrozumabWHO-EMWithdrawnClinical trials