Factor VII

4YT7, 1BF9, 1CVW, 1DAN, 1DVA, 1F7E, 1F7M, 1FAK, 1FF7, 1FFM, 1J9C, 1JBU, 1KLI, 1KLJ, 1O5D, 1QFK, 1W0Y, 1W2K, 1W7X, 1W8B, 1WQV, 1WSS, 1WTG, 1WUN, 1WV7, 1YGC, 1Z6J, 2A2Q, 2AEI, 2AER, 2B7D, 2B8O, 2BZ6, 2C4F, 2EC9, 2F9B, 2FIR, 2FLB, 2FLR, 2PUQ, 2ZP0, 2ZWL, 2ZZU, 3ELA, 3TH2, 3TH3, 3TH4, 4IBL, 4ISH, 4ISI, 4JYU, 4JYV, 4JZD, 4JZE, 4JZF, 4NA9, 4NG9, 4NGA, 4X8S, 4X8T, 4X8U, 4X8V, 4YT6, 4ZXX, 4ZXY, 4Z6A, 4ZMA, 4YLQ, 5I46215514068ENSG00000057593ENSMUSG00000031443P08709P70375NM_000131NM_001267554NM_019616NM_010172NP_000122NP_001254483NP_062562NP_034302Coagulation factor VII (EC 3.4.21.21, formerly known as proconvertin) is a protein involved in coagulation and, in humans, is encoded by gene F7.A biosimilar form of recombinant activated factor VII (AryoSeven) is also available, but does not play any considerable role in the market.The activation of Factor X to Xa initiates the coagulation cascade’s common pathway, leading to clot formation at the site of hemorrhage.Activated FVII binds to endothelial protein C receptor (EPCR), which enhances hemostasis.14 One study showed that eptacog beta binds to EPCR with 25% to 30% more affinity than eptacog alfa, displacing protein C from EPCR binding sites and downregulating activated protein C generation, contributing to its hemostatic effect.[13] Recombinant human factor VII while initially looking promising in intracerebral hemorrhage failed to show benefit following further study and this is no longer recommended.
AliasesHomoloGeneGeneCardsChromosome 13 (human)RNA expressionGene ontologyOrthologsEntrezEnsemblUniProtPubMedWikidataproteincoagulationenzymeserine proteasetissue factorfactor IXfactor Xgenetic recombinationrecombinant factor VIIahemophiliabiosimilarthrombintissue factor pathway inhibitorvitamin Kwarfarinanticoagulantsenzyme cascadefibrinchromosome 13Factor VII deficiencyAryoSevenFactor VIIIIsraeliintracerebral hemorrhageinteractMayer SAMEROPSWayback MachineCoagulation cascadeCoagulation factorsvon Willebrand factor (vWF)Platelet membrane glycoproteinsGlycoprotein Ib (GPIb)Glycoprotein IX (GP9)Glycoprotein IIb/IIIaGPIIIaGlycoprotein VI (GPVI)High-molecular-weight kininogen (HMWK)BradykininPrekallikreinKallikreinFactor XII (Hageman factor)Factor XIFactor III (tissue factor)Factor VProthrombin (factor II)Thrombin (factor IIa)Fibrinogen (factor I)Fibrin (factor Ia)Factor XIIIAnticoagulant factorsAntithrombin (inhibits FII, FIX, FX, FXI, FXII)Protein C (inhibits FV, FVIII)Protein S (cofactor for protein C)Protein Z (inhibits FX)Protein Z-related protease inhibitor (ZPI) (inhibits FX, FXI)Tissue factor pathway inhibitor (TFPI) (inhibits FIII)Fibrinolytic factorsPlasminogenPlasminTissue plasminogen activator (tPA)UrokinasePlasminogen activator inhibitor-1 (PAI-1)Plasminogen activator inhibitor-2 (PAI-2)α2-Antiplasminα2-MacroglobulinThrombin-activatable fibrinolysis inhibitor (TAFI)Coagulation markersPlatelet activationPlatelet factor 4 (PF4)β-Thromboglobulin (β-TG)Thrombin generationProthrombin fragment 1+2 (F1+2)Thrombin–antithrombin complex (TAT)Activated protein C–protein C inhibitor (APC–PCI)Fibrin generationFibrinopeptide A (FpA)Fibrinopeptide B (FpB)Fibrin monomers (FM)FibrinolysisPlasmin-α2-antiplasmin complex (PAP)D-Dimer (DD)Endopeptidasesserine proteases/serine endopeptidasesDigestive enzymesEnteropeptidaseTrypsinChymotrypsinElastaseNeutrophilPancreaticFactor IXaFactor XaFactor XIaFactor XIIaPlasminogen activatorTissue plasminogen activatorUrinary plasminogen activatorComplement systemFactor BFactor DFactor IC3-convertaseimmune systemChymaseGranzymeTryptaseProteinase 3/MyeloblastinVenombinAncrodBatroxobinAcrosinProlyl endopeptidasePronaseProprotein convertasesProstasinReelinSubtilisinSedolisinStreptokinaseCathepsinEnzymesActive siteBinding siteCatalytic triadOxyanion holeEnzyme promiscuityDiffusion-limited enzymeCofactorEnzyme catalysisAllosteric regulationCooperativityEnzyme inhibitorEnzyme activatorEC numberEnzyme superfamilyEnzyme familyList of enzymesEnzyme kineticsEadie–Hofstee diagramHanes–Woolf plotLineweaver–Burk plotMichaelis–Menten kineticsOxidoreductasesTransferasesHydrolasesLyasesIsomerasesLigasesTranslocases